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Tirzepatide

Starting at $369/month*

Powered by dual-action GIP and GLP-1 support, Tirzepatide is clinically proven to curb hunger, accelerate fat loss, improve blood sugar, and reduce inflammation – giving you a powerful edge on your health goals.

*Paid upfront with a 3-month plan. Actual price to the will depend on the plan purchased.

Clinically advanced and provider-guided, Tirzepatide offers dual-action support for appetite control and blood sugar balance - helping you achieve real, sustainable results.

Why Tirzepatide?

Tirzepatide stands out with its dual-action formula—targeting both GIP and GLP-1 receptors—to deliver more powerful results than traditional weight loss medications. By addressing multiple metabolic pathways, it helps regulate appetite, improve insulin function, and support steady, sustainable weight loss.

Accelerates Fat Loss

Targets visceral fat while helping preserve lean muscle mass - ideal for sustainable body recompositing.

Dual Hormone Action

Combines GLP-1 and GIP to improve appetite regulation, glucose control, and insulin response.

Supports Metabolic Longevity

Improves key metabolic markers like blood sugar, inflammation, and cardiovascular health for long-term wellness.

How It Works

“I was able to begin a treatment plan that has helped me lose 40 lbs., and, combined with an existing medication regimen for my diagnoses, has finally seen my blood sugar and hormones balanced. After over a decade of not recognizing the girl in the mirror or photos, my confidence and sense of ownership over my own body have returned in spades! Cannot be more grateful for this place and the abundant care they show their patients. 10/10 HIGHLY and forever will recommend!”

Brittany
Lost 40 lbs

Questions?

We are here to help

What is tirzepatide and how does it support weight loss?

Tirzepatide is a dual GIP and GLP-1 receptor agonist, originally developed to treat type 2 diabetes. It works by targeting two key metabolic pathways that help regulate blood sugar, appetite, and energy balance. For weight loss, tirzepatide reduces hunger, increases fullness, and supports better insulin sensitivity—leading to clinically significant, sustainable results.

Do I need a prescription to get tirzepatide online?

Yes. Tirzepatide is a prescription medication. At ZestRx, every client completes a telehealth consultation and must be approved by a licensed medical provider before starting treatment. This ensures your plan is safe, effective, and tailored to your needs.

Is compounded tirzepatide safe?

When prepared by certified U.S. pharmacies, compounded tirzepatide can be a safe and effective option. ZestRx only sources medications from FDA-registered 503A compounding pharmacies that meet strict quality standards for sterility, potency, and compliance.

What’s the difference between compounded tirzepatide and Mounjaro® or Zepbound®?

Mounjaro® and Zepbound® are brand-name tirzepatide products manufactured by Eli Lilly. Compounded tirzepatide is created by licensed pharmacies and is used when the branded versions are in shortage. While not FDA-approved as standalone products, compounded medications follow regulatory compounding practices and require a prescription. Tirzepatide through ZestRx is also compounded with Niacinamide (Vitamin B3) which can further support weight loss and boost energy levels.

How quickly can I start tirzepatide after my telehealth consult?

Most patients begin treatment within 3–5 business days after approval. Once your provider determines the right dose for you, your medication is shipped directly to your door for convenience and continuity.

What results can I expect with tirzepatide for weight loss?

Results vary by individual, but clinical trials have shown that patients may lose 10–15% of their body weight over time with consistent use, lifestyle support, and proper dosing. Many ZestRx clients also report improved energy, blood sugar control, and reduced cravings as early benefits.

How much does tirzepatide cost per month?

At ZestRx, tirzepatide starts at $399 for your first month with membership. This includes your telehealth consult, ongoing provider check-ins, and medication delivery. Transparent pricing with no hidden fees is part of our promise.

Are there any side effects of tirzepatide?

Some people experience nausea, fatigue, constipation, or GI upset—especially early in treatment. These are usually temporary and can be managed with supportive care and microdosing when needed. ZestRx offers ongoing support and custom titration to help you stay comfortable.

Can I take tirzepatide if I don’t meet the BMI requirement?

We don’t believe BMI tells the whole story. At ZestRx, we look at your overall health, metabolic factors, and weight history—not just a number. Tirzepatide may be appropriate for people managing PCOS, insulin resistance, or other weight-related concerns, regardless of BMI alone.

Is tirzepatide right for me if I have PCOS, insulin resistance, or metabolic issues?

Yes—tirzepatide may be especially helpful for individuals facing these challenges. It improves insulin sensitivity, regulates blood sugar, and supports weight loss—all of which are important for managing PCOS and metabolic dysfunction. Our providers assess your full health profile to determine the best path forward.

How do you ensure the quality of the medications?

ZestRx only partners with licensed U.S. compounding pharmacies that follow strict USP <797> sterile compounding protocols. Each pharmacy is inspected regularly, and all medications are tested for potency, sterility, and purity. We also verify every shipment before it reaches you—so you can feel confident in the care you receive.

Tirzepatide

Clinically advanced and provider-guided, Tirzepatide offers dual-action support for appetite control and blood sugar balance - helping you achieve real, sustainable results.